Macrocyclic peptidomimetics as inhibitors of insulin-regulated aminopeptidase (IRAP)

Barlow, N; Vanga, SR; Savmarker, J; Sandstrom, A; Burns, P; Hallberg, A; Aqvist, J; Gutierrez-de-Teran, H; Hallberg, M; Larhed, M; Chai, SY; Thompson, PE

Thompson, PE (corresponding author), Monash Inst Pharmaceut Sci, Med Chem, Parkville, Vic 3052, Australia.

RSC MEDICINAL CHEMISTRY, 2020; 11 (2): 234

Abstract

Macrocyclic analogues of the linear hexapeptide, angiotensin IV (AngIV) have proved to be potent inhibitors of insulin-regulated aminopeptidase (IRAP,......

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