Lipidated Calcitonin Gene-Related Peptide (CGRP) Peptide Antagonists Retain CGRP Receptor Activity and Attenuate CGRP Action In Vivo

Jamaluddin, A; Chuang, CL; Williams, ET; Siow, A; Yang, SH; Harris, PWR; Petersen, JSSM; Bower, RL; Chand, S; Brimble, MA; Walker, CS; Hay, DL; Loomes, KM

Walker, CS; Hay, DL; Loomes, KM (通讯作者),Univ Auckland, Sch Biol Sci, Auckland, New Zealand.;Hay, DL (通讯作者),Univ Otago, Dept Pharmacol & Toxicol, Dunedin, New Zealand.

FRONTIERS IN PHARMACOLOGY, 2022; 13 ():

Abstract

Signaling through calcitonin gene-related peptide (CGRP) receptors is associated with pain, migraine, and energy expenditure. Small molecule and monoc......

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