Reversible Lysine Specific Demethylase 1 (LSD1) Inhibitors: A Promising Wrench to Impair LSD1

Dai, XJ; Liu, Y; Xue, LP; Xiong, XP; Zhou, Y; Zheng, YC; Liu, HM

Zheng, YC; Liu, HM (corresponding author), Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China.

JOURNAL OF MEDICINAL CHEMISTRY, 2021; 64 (5): 2466

Abstract

As a flavin adenine dinucleotide (FAD)-dependent monoamine oxidase, lysine specific demethylase 1 (LSD1/KDM1A) functions as a transcription coactivato......

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