Multi-step virtual screening to develop selective DYRK1A inhibitors

Koyama, T; Yamaotsu, N; Nakagome, I; Ozawa, S; Yoshida, T; Hayakawa, D; Hirono, S

Koyama, T; Hirono, S (reprint author), Kitasato Univ, Sch Pharm, Minato Ku, 5-9-1 Shirokane, Tokyo 1088641, Japan.

JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2017; 72 ( ): 229

Abstract

Developing selective inhibitors for a particular kinase remains a major challenge in kinase-targeted drug discovery. Here we performed a multi-step vi......

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