Tofacitinib Synthesis - An Asymmetric Challenge

Carvalho, LCR; Lourenco, A; Ferreira, LM; Branco, PS

Carvalho, LCR (reprint author), Univ Nova Lisboa, Fac Ciancias & Tecnol, Dept Quim, P-2829516 Caparica, Portugal.

EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2019; 2019 (4): 615

Abstract

Tofacitinib is a Janus activated kinase (JAK) inhibitor approved for the treatment of rheumatoid arthritis and active psoriatic arthritis. Its synthes......

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