BET bromodomain inhibitors

Schwalm, MP; Knapp, S

Knapp, S (通讯作者),Goethe Univ Frankfurt, Inst Pharmazeut Chem, Biozentrum, Max Von Laue Str 9, D-60438 Frankfurt, Germany.;Knapp, S (通讯作者),Goethe Univ Frankfurt, Buchmann Inst Life Sci, Struct Genom Consortium, Max Von Laue Str 15, D-60438 Frankfurt, Germany.;Knapp, S (通讯作者),German Canc Res Ctr, German Canc Consortium DKTK, DKTK Site Frankfurt Mainz, D-69120 Heidelberg, Germany.

CURRENT OPINION IN CHEMICAL BIOLOGY, 2022; 68 ():

Abstract

Lysine acetylation creates docking sites for epigenetic reader domains of BET bromodomain proteins that have emerged as principal regulators of linage......

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