Hot-spot guided design of macrocyclic inhibitors of the LSD1-CoREST1 interaction

Hart, P; Openy, J; Krzyzanowski, A; Adihou, H; Waldmann, H

Waldmann, H (reprint author), Max Planck Inst Mol Physiol, Dept Chem Biol, Otto Hahn Str 11, D-44227 Dortmund, Germany.

TETRAHEDRON, 2019; 75 (48):

Abstract

New modalities such as cyclic peptides are attractive structures to inhibit challenging targets. The interaction between LSD1 and CoREST1 is required ......

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