KSQ-4279, a first-in-class USP1 inhibitor shows strong combination activity in BRCA mutant cancers with intrinsic or acquired resistance to PARP inhibitors

Cadzow, L; Gokhale, PC; Ganapathy, S; Sullivan, P; Nayak, S; Shenker, S; Schlabach, M; Tobin, E; Matulonis, UA; Liu, JF; Stegmeier, F; Wylie, A

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