期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (7)
A regioselective C-H functionalization/annulation reaction of N-sulfonyl amides and allylbenzenes through a palladium-catalyzed C(sp(2))-H allylation/......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (8)
A novel protocol for the synthesis of pyrido[2,3-b]indoles (alpha-carbolines, 3) from (E)-3-(2-oxo-2-phenylethylidene) indolin-2-one derivatives 1 and......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (11)
Herein we describe a catalyst-free regioselective [3 + 3] annulation/oxidation reaction of cyclic amidines such as DBU (1,8-diazabicyclo(5.4.0)undec-7......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (12)
A visible-light-driven photoredox reaction of tetrahydroisoquinoline with 2H-azirines is described. 4,7-Bis(4-methoxyphenyl)benzo[ c][1,2,5]thiadiazol......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (12)
A facile and effective synthesis of 2-chloromethylpyridines was developed by a one-pot reaction of 2-alkylpyridin-Noxides and triphosgene at room temp......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (12)
Iodine(III)-mediated synthesis of 4-iodo-N-phenylaniline from iodobenzene has been achieved, and the reaction can proceed under mild conditions. A var......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (12)
Tetrathiatriarylmethyl (trityl) radicals have been recently shown to react with biological oxidoreductants including glutathione (GSH), ascorbic acid ......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (13)
An operationally simple synthesis of Z-configured and C3-unsubstituted N-sulfonyl- 2-iminocoumarins (e.g., 8a) that proceeds under mild conditions is ......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (13)
1,3-Dipolar cycloaddition of azomethine ylides and electron deficient alkenes is widely studied for rapid installation of pyrrolidine frameworks. Desp......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (14)
Herein, we present a novel silver- or copper-mediated direct amidation-ketonization-selenation of terminal allcynes for the synthesis of alpha-oxo-sel......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (15)
A diversity-oriented chemoenzymatic approach for the collective preparation of sulfated core 2 O-GalNAc glycans and their nonsulfated counterparts was......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (16)
Inactivation of the flavoenzyme-encoding gene flsO1 in fluostatin biosynthesis led to the isolation of four new angucyclinone derivatives (11, 12, 14,......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (8)
A novel route for ortho-selective C-H borylation of 2-phenylthiopyridines using BBr3 as the boron source under metal-free conditions has been reported......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (9)
A novel copper-catalyzed cyclization of readily available vinyl azides with CF3-ynones is steadily achieved under mild conditions to furnish the versa......
期刊: JOURNAL OF ORGANIC CHEMISTRY, 2021; 86 (11)
A metal-free intramolecular [3+2] cycloaddtion has been achieved by treating benzene-linked propynol-ynes with AcOH/H2O in a one-pot manner. The react......